SCHEMBL4785519

SCHEMBL4785519

CC(C)(C)OC(=O)CC(NC(=O)c1cnc2cc(C(F)(F)F)ccc2c1N1CCSCC1)C(O)CF

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.44
DPP4 P27487 1/20 0.33
MMP1 P03956 2/20 0.33
MMP9 P14780 2/20 0.33
MMP13 P45452 2/20 0.33
PDGFRB P09619 1/20 0.32
CYP8B1 Q9UNU6 3/20 0.32
MET P08581 1/20 0.32
ADAM17 P78536 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4742128 0.92 THRB (0.45) THRBCYP8B1
SCHEMBL4743466 0.91 THRB (0.46) THRB
SCHEMBL4742105 0.90 THRB (0.45) THRBPDGFRBCYP8B1MET
SCHEMBL4785468 0.88 THRB (0.45) THRBDPP4MMP1MMP9MMP13
SCHEMBL4785514 0.81 THRB (0.46) THRBDPP4MMP1MMP9MMP13
SCHEMBL4741630 0.80 THRB (0.46) THRBMMP1MMP9MMP13CYP8B1
SCHEMBL4743062 0.79 THRB (0.47) THRB
SCHEMBL4742589 0.78 MET (0.44) THRBPDGFRBMET
SCHEMBL4742145 0.77 THRB (0.43) THRBDPP4MMP1MMP9MMP13
Trifluoroacetic Acid SCHEMBL4742140 0.76 THRB (0.43) THRBDPP4MMP1MMP9MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed