SCHEMBL4739339

SCHEMBL4739339

CC(C)(C)OC(=O)CC(NC(=O)c1cnc2cc([N+](=O)[O-])ccc2c1N1CCN(C(=O)OC(C)(C)C)CC1)C(=O)CF

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MET P08581 9/20 0.46
MAPT P10636 3/20 0.45
ALDH1A1 P00352 2/20 0.45
LMNA P02545 2/20 0.45
KCNH2 Q12809 4/20 0.35
PTPN11 Q06124 1/20 0.35
THRB P10828 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
MEN1 O00255 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
CCNT1 O60563 1/20 0.34
CDK9 P50750 1/20 0.34
KIT P10721 2/20 0.34
PDGFRB P09619 2/20 0.34
PDGFRA P16234 1/20 0.34
FLT3 P36888 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4785479 0.89 THRB (0.42) METMAPTALDH1A1LMNAPTPN11
SCHEMBL4742589 0.88 MET (0.44) METMAPTALDH1A1LMNAKCNH2
SCHEMBL4743406 0.85 MET (0.39) METMAPTALDH1A1LMNAPTPN11
SCHEMBL4742143 0.80 ALDH1A1 (0.58) METMAPTALDH1A1LMNAKCNH2
SCHEMBL4743037 0.80 MAPT (0.40) MAPTLMNAPTPN11THRBKIT
SCHEMBL4742118 0.80 MET (0.38) METMAPTALDH1A1LMNATHRB
SCHEMBL4742621 0.79 USP2 (0.45) METMAPTLMNAPTPN11SMN1; SMN2
SCHEMBL4785468 0.79 THRB (0.45) METTHRB
SCHEMBL4743062 0.79 THRB (0.47) MAPTALDH1A1THRBSMN1; SMN2TSHR
SCHEMBL4742104 0.79 MAPT (0.53) METMAPTALDH1A1LMNATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed