SCHEMBL4741747

SCHEMBL4741747

COc1ccc(C(=O)Nc2sc(-c3ccccc3)nc2-c2ccccc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.65
NPC1 O15118 1/20 0.65
RAB9A P51151 1/20 0.65
KMT2A Q03164 1/20 0.65
RXFP1 Q9HBX9 1/20 0.65
ADORA1 P30542 7/20 0.63
KDM4E B2RXH2 2/20 0.62
ALDH1A1 P00352 1/20 0.62
MAPT P10636 1/20 0.62
ADORA3 P0DMS8 11/20 0.61
PTGDR2 Q9Y5Y4 2/20 0.57
ADORA2A P29274 2/20 0.57
CSNK2A2 P19784 1/20 0.54
CSNK2A1 P68400 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4738310 0.87 ALDH1A1 (0.71) NPC1RAB9AKMT2AADORA1KDM4E
SCHEMBL4737640 0.84 KDM4E (0.63) MEN1NPC1RAB9AKMT2ARXFP1
SCHEMBL14148529 0.82 KDM4E (0.58) MEN1NPC1RAB9AKMT2ARXFP1
SCHEMBL4737628 0.82 KDM4E (0.64) KDM4EALDH1A1MAPT
SCHEMBL4737623 0.81 KDM4E (0.60) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL235277 0.79 ADORA1 (0.78) MEN1NPC1RAB9AKMT2ARXFP1
SCHEMBL14148658 0.79 LMNA (0.76) MEN1NPC1RAB9AKMT2AADORA1
SCHEMBL6436649 0.78 MAPT (0.53) MEN1NPC1RAB9AKMT2AKDM4E
SCHEMBL977661 0.78 CDC7 (0.70) MEN1NPC1RAB9AKMT2ARXFP1
SCHEMBL4268936 0.77 KDM4E (0.77) MEN1KMT2AKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008090382-A1 THIAZOLE AND OXAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PRION DISEASES, CANCER AND CONDITIONS OF THE CENTRAL NERVOUS SYSTEM AS WELL AS IN THE REGULATION OF STEM CELLS THE UNIVERSITY OF SHEFFIELD (GB) 2008-07-31 WO disclosed
WO-2008090382-A1 THIAZOLE AND OXAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PRION DISEASES, CANCER AND CONDITIONS OF THE CENTRAL NERVOUS SYSTEM AS WELL AS IN THE REGULATION OF STEM CELLS THE UNIVERSITY OF SHEFFIELD (GB) 2008-07-31 WO disclosed