SCHEMBL4741778

SCHEMBL4741778

COC(=O)c1cccc(CCO[Si](C)(C)C(C)(C)C)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 3/20 0.59
CYP4A11 Q02928 3/20 0.59
LOXL2 Q9Y4K0 1/20 0.54
SLC7A5 Q01650 1/20 0.47
MRGPRX4 Q96LA9 2/20 0.46
ABHD6 Q9BV23 1/20 0.46
PARP1 P09874 1/20 0.45
TSHR P16473 1/20 0.45
FOLH1 Q04609 1/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 1/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
HIF1A Q16665 1/20 0.43
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21068861 0.92 CYP4F2 (0.60) CYP4F2CYP4A11LOXL2SLC7A5MRGPRX4
SCHEMBL4876076 0.86 MAOB (0.43) CYP4F2CYP4A11SLC7A5MRGPRX4HPGD
SCHEMBL4741394 0.86 FOLH1 (0.46) CYP4F2CYP4A11MRGPRX4FOLH1ALDH1A1
SCHEMBL8320447 0.86 LOXL2 (0.56) CYP4F2CYP4A11LOXL2SLC7A5MRGPRX4
SCHEMBL18579747 0.82 CYP4F2 (0.43) CYP4F2CYP4A11LOXL2TSHRALDH1A1
SCHEMBL7241207 0.81 ATAD2 (0.41) CYP4F2CYP4A11LOXL2SLC7A5ABHD6
SCHEMBL10145035 0.81 MAPT (0.49) MRGPRX4ALDH1A1NPC1KMT2ASMN1; SMN2
SCHEMBL15019978 0.80 CYP4F2 (0.73) CYP4F2CYP4A11LOXL2SLC7A5MRGPRX4
SCHEMBL31126580 0.80 LOXL2 (0.43) CYP4F2CYP4A11LOXL2SLC7A5MRGPRX4
SCHEMBL70173 0.80 CYP4F2 (0.83) CYP4F2CYP4A11LOXL2SLC7A5MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3901156-A1 NITROOXYDERIVATIVE OF ROCK KINASE INHIBITOR Vivavision (Shanghai) Ltd (CN) 2021-10-27 EP disclosed
WO-2008096129-A1 NITROGEN CONTAINING HETROCYCLIC COMPOUNDS USEFUL AS BIFUNCTIONAL MODULATORS OF M3 RECEPTORS AND BETA- 2 RECEPTORS ARGENTA DISCOVERY LTD (GB) 2008-08-14 WO disclosed