SCHEMBL4742560

SCHEMBL4742560

O=S(=O)(CCCBr)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 1/20 0.52
KEAP1 Q14145 1/20 0.51
NFE2L2 Q16236 1/20 0.51
HDAC1 Q13547 2/20 0.50
HDAC8 Q9BY41 2/20 0.50
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50
HDAC11 Q96DB2 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
HDAC9 Q9UKV0 1/20 0.50
HDAC5 Q9UQL6 1/20 0.50
HSD11B1 P28845 5/20 0.48
MMP3 P08254 2/20 0.47
MMP8 P22894 2/20 0.47
MMP13 P45452 2/20 0.47
MMP1 P03956 1/20 0.47
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6096865 0.94 KEAP1 (0.54) PSIP1KEAP1NFE2L2HDAC1HDAC8
SCHEMBL7744005 0.92 HDAC1 (0.56) PSIP1KEAP1NFE2L2HDAC1HDAC8
SCHEMBL9672257 0.89 ALDH1A1 (0.58) KEAP1NFE2L2HDAC1HDAC8HDAC3
SCHEMBL1779667 0.86 PSIP1 (0.56) PSIP1KEAP1NFE2L2HDAC1HDAC8
SCHEMBL10629823 0.86 PSIP1 (0.61) PSIP1KEAP1NFE2L2HDAC1HDAC8
SCHEMBL576918 0.86 KEAP1 (0.63) PSIP1KEAP1NFE2L2HDAC1HDAC8
SCHEMBL10626503 0.84 HDAC1 (0.65) PSIP1KEAP1NFE2L2HDAC1HDAC8
SCHEMBL777601 0.81 PSIP1 (0.67) PSIP1KEAP1NFE2L2HDAC1HDAC8
SCHEMBL5387555 0.81 PLCG1 (0.59) HSD11B1ALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL8972497 0.80 PSIP1 (0.54) PSIP1KEAP1NFE2L2HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016014426-A1 ORGANIC REACTIONS THE ARIZONA BOARD OF REGENTS (US) 2016-01-28 WO disclosed
CN-103509135-B Olefin polymerization catalyst component, preparation method and application thereof CHINA PETROLEUM & CHEMICAL 2015-07-22 CN disclosed
CN-101252929-A G protein-coupled receptor agonists PROSIDION LTD (GB) 2008-08-27 CN disclosed
WO-2008096128-A1 OXAZOLE AND THIAZOLE DERIVATIVES AND THEIR USES 2 ARGENTA DISCOVERY LTD (GB) 2008-08-14 WO disclosed
US-6051605-A TREATING PSYCHOSIS AND SCHIZOPHRENIA USING A COMPOUND THAT IS AN ANTAGONIST OF DOPAMINE D4 RECEPTORS WARNER-LAMBERT COMPANY (US) 2000-04-18 US disclosed
US-4775674-A CARDIOTONIC AGENTS BRISTOL-MYERS COMPANY (US) 1988-10-04 US disclosed