SCHEMBL4743037

SCHEMBL4743037

CC(C)(C)OC(=O)CC(NC(=O)c1cnc2c(F)cccc2c1N1CCN(C(=O)OC(C)(C)C)CC1)C(=O)CF

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.40
PTPN11 Q06124 1/20 0.39
ACHE P22303 1/20 0.37
GPR119 Q8TDV5 2/20 0.37
CKS1B P61024 1/20 0.37
SKP1 P63208 1/20 0.37
SKP2 Q13309 1/20 0.37
GBA1 P04062 1/20 0.36
TP53 P04637 2/20 0.36
THRB P10828 1/20 0.36
KIT P10721 1/20 0.36
BACE1 P56817 1/20 0.36
CXCR2 P25025 1/20 0.35
USP2 O75604 1/20 0.35
MAPK1 P28482 1/20 0.35
RECQL P46063 1/20 0.35
HSD17B10 Q99714 1/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
GLA P06280 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4742621 0.92 USP2 (0.45) MAPTPTPN11ACHECKS1BSKP1
SCHEMBL4743406 0.90 MET (0.39) MAPTPTPN11ACHECKS1BSKP1
SCHEMBL4785479 0.85 THRB (0.42) MAPTPTPN11GPR119CKS1BSKP1
SCHEMBL4739339 0.80 MET (0.46) MAPTPTPN11THRBKITLMNA
SCHEMBL4743456 0.80 MAPT (0.47) MAPTPTPN11ACHEGPR119CKS1B
SCHEMBL4742558 0.79 USP2 (0.44) MAPTPTPN11ACHECKS1BSKP1
SCHEMBL4743039 0.79 USP2 (0.35) MAPTTP53USP2MAPK1RECQL
SCHEMBL4741642 0.78 MAPT (0.64) MAPTTP53USP2MAPK1RECQL
SCHEMBL4786909 0.77 MET (0.39) MAPTPTPN11ACHETP53BACE1
SCHEMBL4785468 0.72 THRB (0.45) THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed