SCHEMBL4743259

SCHEMBL4743259

Cc1cc(C(=O)c2ccc(Cl)cc2)c(C)c(C)c1OCCCCCN1CCN(CC(=O)NC(C)C)CC1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 6/20 0.43
KCNA5 P22460 1/20 0.40
HRH3 Q9Y5N1 7/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
ATM Q13315 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HTR1A P08908 1/20 0.39
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4744714 0.90 AVPR1B (0.46) AVPR1BKCNA5HRH3SMN1; SMN2KDM4E
SCHEMBL4744692 0.86 KDM4E (0.51) AVPR1BKCNA5HRH3SMN1; SMN2KDM4E
SCHEMBL4743105 0.85 AVPR1B (0.44) AVPR1BKCNA5HRH3HTR1AHTR2A
SCHEMBL4743288 0.82 HRH3 (0.56) KCNA5HRH3
SCHEMBL4743111 0.82 HRH3 (0.56) KCNA5HRH3
SCHEMBL4745354 0.82 HRH3 (0.37) AVPR1BHRH3ATM
SCHEMBL4743293 0.81 MEN1 (0.56) KCNA5HRH3KDM4E
SCHEMBL4745334 0.81 HRH3 (0.47) AVPR1BKCNA5HRH3
SCHEMBL4745400 0.81 HTR1A (0.50) AVPR1BKCNA5HRH3HTR1AHTR2A
SCHEMBL4743291 0.81 HRH3 (0.48) AVPR1BKCNA5HRH3HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008107320-A1 PIPERIDINE AND PIPERAZINE DERIVATIVES USED AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO disclosed