SCHEMBL4743443

SCHEMBL4743443

O=C(O)c1cnc2cc(C(F)(F)F)ccc2c1N1CCSCC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.53
DPP4 P27487 1/20 0.41
POLB P06746 1/20 0.40
CYP8B1 Q9UNU6 3/20 0.40
ADRB2 P07550 1/20 0.40
NCF1 P14598 1/20 0.40
LIPG Q9Y5X9 1/20 0.39
CSF1R P07333 1/20 0.38
SCN10A Q9Y5Y9 1/20 0.38
PLK4 O00444 1/20 0.38
DYRK3 O43781 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
CHEK2 O96017 1/20 0.38
FGFR1 P11362 1/20 0.38
CDK2 P24941 1/20 0.38
FLT4 P35916 1/20 0.38
KDR P35968 1/20 0.38
CLK2 P49760 1/20 0.38
GSK3A P49840 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4743041 0.88 THRB (0.55) THRBCYP8B1ADRB2NCF1LIPG
SCHEMBL4743063 0.86 THRB (0.56) THRBALDH1A1SMN1; SMN2HSD17B10
SCHEMBL4742585 0.84 THRB (0.75) THRBALDH1A1HSD17B10
SCHEMBL4739993 0.80 THRB (0.54) THRBCYP8B1SMN1; SMN2HPGD
Trifluoroacetic Acid SCHEMBL4742140 0.79 THRB (0.43) THRBDPP4CYP8B1SCN10AALDH1A1
SCHEMBL4785514 0.75 THRB (0.46) THRBDPP4CYP8B1ADRB2NCF1
SCHEMBL3887756 0.75 ALDH1A1 (0.46) THRBCSF1RPLK4DYRK3PRKD3
SCHEMBL30592902 0.75 ALDH1A1 (0.46) THRBCSF1RPLK4DYRK3PRKD3
SCHEMBL4785468 0.75 THRB (0.45) THRBDPP4CYP8B1SCN10A
Hydrochloric Acid SCHEMBL11870232 0.74 ALDH1A1 (0.45) THRBCSF1RPLK4DYRK3PRKD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed