SCHEMBL4785514

SCHEMBL4785514

CC(O)C(NC(=O)c1cnc2cc(C(F)(F)F)ccc2c1N1CCSCC1)C(F)C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.46
DPP4 P27487 1/20 0.34
PDGFRB P09619 1/20 0.33
CYP8B1 Q9UNU6 4/20 0.33
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
MMP13 P45452 1/20 0.32
PDE6D O43924 1/20 0.32
PDE5A O76074 1/20 0.32
PDE6A P16499 1/20 0.32
PDE6G P18545 1/20 0.32
PDE6B P35913 1/20 0.32
PDE6C P51160 1/20 0.32
PDE6H Q13956 1/20 0.32
SCN10A Q9Y5Y9 1/20 0.32
MET P08581 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
ADRB2 P07550 1/20 0.31
NCF1 P14598 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4785519 0.81 THRB (0.44) THRBDPP4PDGFRBCYP8B1MMP1
SCHEMBL4785468 0.81 THRB (0.45) THRBDPP4CYP8B1MMP1MMP9
SCHEMBL4743443 0.75 THRB (0.53) THRBDPP4CYP8B1SCN10AADRB2
SCHEMBL4742585 0.75 THRB (0.75) THRBPDE6DPDE5APDE6APDE6G
Trifluoroacetic Acid SCHEMBL4742140 0.73 THRB (0.43) THRBDPP4CYP8B1MMP1MMP9
SCHEMBL4742145 0.73 THRB (0.43) THRBDPP4PDGFRBCYP8B1MMP1
SCHEMBL4742128 0.73 THRB (0.45) THRBCYP8B1MAPT
SCHEMBL4741630 0.72 THRB (0.46) THRBCYP8B1MMP1MMP9MMP13
SCHEMBL4743466 0.72 THRB (0.46) THRBMAPT
SCHEMBL4743062 0.71 THRB (0.47) THRBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed