SCHEMBL4743715

SCHEMBL4743715

O=C(c1cncc(OC2CCN(C(=O)O)CC2)c1)c1ncc[nH]1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
HTT P42858 1/20 0.41
CYP11B2 P19099 2/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
PRMT5 O14744 1/20 0.37
OPRK1 P41145 1/20 0.36
KCNH2 Q12809 1/20 0.36
EPHX2 P34913 1/20 0.36
HTR2B P41595 1/20 0.35
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
GSK3B P49841 1/20 0.35
NAMPT P43490 1/20 0.35
RIPK2 O43353 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4786833 0.74 ALDH1A1 (0.44) ALDH1A1HTTCYP11B2PRMT5OPRK1
SCHEMBL17555503 0.73 L3MBTL4 (0.43) ALDH1A1HTTCYP11B2EPHX2
SCHEMBL19473362 0.69 PRMT5 (0.45) ALDH1A1HTTCYP11B2PRMT5OPRK1
SCHEMBL2305909 0.69 EPHX2 (0.63) ALDH1A1HTTEPHX2
SCHEMBL17559499 0.68 PRMT5 (0.44) ALDH1A1HTTCYP11B2PRMT5OPRK1
SCHEMBL639198 0.68 EPHX2 (0.60) ALDH1A1HTTEPHX2NAMPT
SCHEMBL28886445 0.67 HTT (0.51) ALDH1A1HTTNPC1RAB9A
SCHEMBL1117853 0.67 RAB9A (0.62) ALDH1A1HTTNPC1RAB9ANAMPT
SCHEMBL17559339 0.67 PRMT5 (0.45) ALDH1A1HTTCYP11B2PRMT5EPHX2
SCHEMBL4745663 0.67 GPR119 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008109613-A1 BENZO[C][2,7]NAPHTHYRIDINE DERIVATIVES, AND THEIR USE AS KINASE INHIBITORS WYETH (US) 2008-09-12 WO disclosed