SCHEMBL474455

SCHEMBL474455

CC(c1cc(C(=O)O)ccc1-c1ccccc1)C(O)(c1cc(F)c2c(c1)N(C)C(=O)CO2)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.32
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31
MALT1 Q9UDY8 1/20 0.31
HTR1A P08908 1/20 0.30
HTR1D P28221 1/20 0.30
HTR1B P28222 1/20 0.30
S1PR1 P21453 1/20 0.30
TTR P02766 1/20 0.30
HPSE Q9Y251 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474611 0.92 SMN1; SMN2 (0.35) ALDH1A1MALT1HTR1AHTR1DHTR1B
SCHEMBL473958 0.87 ALDH1A1 (0.37) ALDH1A1LMNAMALT1
SCHEMBL474375 0.85 ALDH1A1 (0.37) ALDH1A1LMNAAKR1C3AKR1C2HTR1A
SCHEMBL474394 0.80 POLB (0.36) ALDH1A1MALT1
SCHEMBL474658 0.77 SMN1; SMN2 (0.36) ALDH1A1
SCHEMBL474282 0.77 MALT1 (0.33) MALT1
SCHEMBL12163875 0.77 MALT1 (0.33) MALT1
SCHEMBL474476 0.76 MAPK14 (0.35)
SCHEMBL474660 0.75 MALT1 (0.32) MALT1
SCHEMBL473939 0.75 BDKRB1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed