SCHEMBL474375

SCHEMBL474375

CC(c1cc(C(=O)O)ccc1-c1ccccc1)C(O)(c1cccc2c1OCC(=O)N2C)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
AKR1C3 P42330 2/20 0.34
AKR1C2 P52895 2/20 0.34
LMNA P02545 1/20 0.33
TTR P02766 1/20 0.33
S1PR1 P21453 1/20 0.33
PDCD1 Q15116 2/20 0.33
CD274 Q9NZQ7 2/20 0.33
CMA1 P23946 1/20 0.32
SRD5A2 P31213 1/20 0.32
PRKAG1 P54619 1/20 0.31
PRKAA1 Q13131 1/20 0.31
PRKAB1 Q9Y478 1/20 0.31
HPSE Q9Y251 2/20 0.31
RECQL P46063 1/20 0.31
HSD17B10 Q99714 1/20 0.31
RIPK1 Q13546 1/20 0.30
HTR1A P08908 1/20 0.30
HTR1D P28221 1/20 0.30
HTR1B P28222 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474658 0.92 SMN1; SMN2 (0.36) ALDH1A1PDCD1CD274HSD17B10CCKBR
SCHEMBL474455 0.85 ALDH1A1 (0.34) ALDH1A1AKR1C3AKR1C2LMNATTR
SCHEMBL473958 0.84 ALDH1A1 (0.37) ALDH1A1LMNARIPK1NR1H2NR1H3
SCHEMBL474611 0.78 SMN1; SMN2 (0.35) ALDH1A1HTR1AHTR1DHTR1B
SCHEMBL474476 0.78 MAPK14 (0.35)
SCHEMBL12163900 0.77 RORC (0.35) CMA1
SCHEMBL474394 0.76 POLB (0.36) ALDH1A1HSD17B10
SCHEMBL474404 0.76 MALT1 (0.34) HTR1AHTR1DHTR1BSLC6A4KCNH2
SCHEMBL15520787 0.74 MALT1 (0.33) HTR1AHTR1DHTR1B
SCHEMBL474520 0.74 BDKRB1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed