SCHEMBL4745351

SCHEMBL4745351

Cc1cc(C2(C)CC2)ccc1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
POLB P06746 1/20 0.40
CASP6 P55212 1/20 0.40
BACE1 P56817 1/20 0.36
ESR1 P03372 2/20 0.36
ESR2 Q92731 2/20 0.36
DAPK3 O43293 1/20 0.36
NTRK1 P04629 1/20 0.36
PIM1 P11309 1/20 0.36
FLT3 P36888 1/20 0.36
GSK3B P49841 1/20 0.36
ROCK1 Q13464 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
KCNJ6 P48051 1/20 0.34
KCNJ5 P48544 1/20 0.34
KCNJ3 P48549 1/20 0.34
ACHE P22303 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12898001 0.83 AKR1B10 (0.45) HDAC1HDAC6BACE1ESR1ESR2
SCHEMBL14625259 0.83 SLC6A3 (0.47) HDAC3HDAC1HDAC2HDAC6BACE1
SCHEMBL14625193 0.78 SLC6A3 (0.51) HDAC3HDAC1HDAC2HDAC6POLB
SCHEMBL24746321 0.78 ABCC9 (0.36) SLC6A3SLC6A2SLC6A4IDO1
SCHEMBL1905906 0.78 SLC6A4 (0.36) ESR2SLC6A3SLC6A2SLC6A4
SCHEMBL8418296 0.78 POLB (0.45) HDAC3HDAC1HDAC2HDAC6POLB
SCHEMBL26607109 0.75 ESR1 (0.36) POLBESR1ESR2ACHECCR2
SCHEMBL257534 0.75 SLC6A3 (0.49) HDAC3HDAC1HDAC2HDAC6SLC6A3
SCHEMBL19507134 0.75 SMN1; SMN2 (0.44) HDAC3HDAC1HDAC2HDAC6POLB
SCHEMBL24746227 0.75 HDAC3 (0.49) HDAC3HDAC1HDAC2HDAC6POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022174253-A1 HPK1 ANTAGONISTS AND USES THEREOF Nimbus Saturn, Inc. (US) 2022-08-18 WO disclosed
WO-2017006283-A1 DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CONTAINING CYCLOPROPANO LINKAGE CV6 THERAPEUTICS (NI) LIMITED (GB) 2017-01-12 WO disclosed
WO-2008104101-A1 1-(3-METHYL-4-FLUORO) PHENYL-1-METHYLCYCLOPROPANE COMPOUNDS AND USE THEREOF SINOCHEM CORPORATION (CN) 2008-09-04 WO disclosed
WO-2008104101-A1 1-(3-METHYL-4-FLUORO) PHENYL-1-METHYLCYCLOPROPANE COMPOUNDS AND USE THEREOF SINOCHEM CORPORATION (CN) 2008-09-04 WO disclosed
WO-2005103055-A1 PYRAZOLO-[4,3-e]-1,2,4-TRIAZOLO-[1,5-c]-PYRIMIDINE ADENOSINE A2A RECEPTOR ANTAGONISTS SCHERING CORPORATION (US) 2005-11-03 WO disclosed