SCHEMBL4745393

SCHEMBL4745393

O=S(=O)(c1ccc(Sc2ccccn2)c2nonc12)N1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.45
COMT P21964 2/20 0.43
TSHR P16473 4/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
ALDH1A1 P00352 7/20 0.41
HTT P42858 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
LMNA P02545 2/20 0.39
MCOLN3 Q8TDD5 1/20 0.39
POLB P06746 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PKM P14618 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4787284 0.84 TSHR (0.52) KDM4ETSHRCYP2C19ALDH1A1HTT
SCHEMBL4787718 0.83 TSHR (0.41) KDM4ETSHRALDH1A1HTTNPSR1
SCHEMBL4787514 0.83 L3MBTL1 (0.52) KDM4ECOMTTSHRALDH1A1HTT
SCHEMBL4746814 0.82 TP53 (0.43) COMTTSHRALDH1A1HTTMEN1
SCHEMBL4816303 0.81 CCR1 (0.46) TSHRALDH1A1HTTMEN1KMT2A
SCHEMBL4745419 0.78 MCOLN3 (0.46) KDM4ETSHRCYP3A4CYP2C9CYP2C19
SCHEMBL4746866 0.75 HTT (0.48) KDM4ETSHRALDH1A1HTTMEN1
SCHEMBL4745397 0.74 KMT2A (0.43) CYP3A4CYP2C19ALDH1A1MEN1KMT2A
SCHEMBL5244145 0.72 L3MBTL1 (0.50) TSHRALDH1A1KMT2AL3MBTL1PKM
SCHEMBL5242720 0.72 ALDH1A1 (0.67) TSHRALDH1A1HTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008115259-A2 DERIVATIVES OF BENZOXADIAZOLE SUITABLE FOR THE TREATMENT OF CELL PROLIFERATIVE DISEASES RIGEL PHARMACEUTICALS, INC. (US) 2008-09-25 WO claimed