SCHEMBL474633

SCHEMBL474633

CC(c1cc(C(=O)O)ccc1-c1ccccc1)C(O)(c1ccc2c(c1)n(C)c(=O)n2C)C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
GLA P06280 1/20 0.41
HTT P42858 1/20 0.36
MAPK14 Q16539 2/20 0.36
BRPF1 P55201 4/20 0.36
KDM4E B2RXH2 2/20 0.36
BRD4 O60885 2/20 0.36
HSD17B10 Q99714 1/20 0.36
S1PR1 P21453 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
CMA1 P23946 1/20 0.35
GAA P10253 1/20 0.35
PRKAG1 P54619 1/20 0.34
PRKAA1 Q13131 1/20 0.34
PRKAB1 Q9Y478 1/20 0.34
PGR P06401 1/20 0.33
NR1H3 Q13133 1/20 0.33
TTR P02766 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473904 0.86 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2AKR1C3AKR1C2
SCHEMBL474051 0.85 ALDH1A1 (0.39) ALDH1A1S1PR1PRKAG1PRKAA1PRKAB1
SCHEMBL474933 0.84 PPARG (0.39) ALDH1A1SMN1; SMN2BRPF1KDM4EBRD4
SCHEMBL474247 0.83 TNKS2 (0.39) ALDH1A1SMN1; SMN2GLABRPF1KDM4E
SCHEMBL12163997 0.83 TNKS2 (0.39) ALDH1A1SMN1; SMN2GLABRPF1KDM4E
SCHEMBL474508 0.82 SRD5A2 (0.41) ALDH1A1SMN1; SMN2GLABRPF1KDM4E
SCHEMBL474443 0.81 AKR1C3 (0.37) ALDH1A1SMN1; SMN2GLABRPF1AKR1C3
SCHEMBL12163978 0.81 AKR1C3 (0.37) ALDH1A1SMN1; SMN2GLABRPF1AKR1C3
SCHEMBL474483 0.81 SMN1; SMN2 (0.35) ALDH1A1SMN1; SMN2GLAMAPK14BRPF1
SCHEMBL474521 0.81 TP53 (0.39) ALDH1A1SMN1; SMN2GLAHTTMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed