SCHEMBL474483

SCHEMBL474483

CC(c1c(-c2ccccc2)ccc(F)c1C(=O)O)C(O)(c1ccc2c(c1)n(C)c(=O)n2C)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 1/20 0.35
GLA P06280 1/20 0.35
MAPK14 Q16539 2/20 0.35
AKR1C3 P42330 4/20 0.35
AKR1C2 P52895 4/20 0.35
PTGS1 P23219 3/20 0.35
MEN1 O00255 2/20 0.35
PTGS2 P35354 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPT P10636 2/20 0.35
FABP2 P12104 1/20 0.35
TSHR P16473 1/20 0.35
AKR1C4 P17516 1/20 0.35
ADRA2B P18089 1/20 0.35
CHRM3 P20309 1/20 0.35
HTR2C P28335 1/20 0.35
DRD3 P35462 1/20 0.35
AKR1C1 Q04828 1/20 0.35
SLC22A6 Q4U2R8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474521 0.85 TP53 (0.39) SMN1; SMN2ALDH1A1GLAMAPK14GAA
SCHEMBL474633 0.81 ALDH1A1 (0.41) SMN1; SMN2ALDH1A1GLAMAPK14AKR1C3
SCHEMBL474975 0.81 ALDH1A1 (0.35) SMN1; SMN2ALDH1A1GLAMAPK14PTGS1
SCHEMBL474933 0.75 PPARG (0.39) SMN1; SMN2ALDH1A1MEN1KMT2AMAPT
SCHEMBL474508 0.73 SRD5A2 (0.41) SMN1; SMN2ALDH1A1GLAAKR1C3AKR1C2
SCHEMBL12163970 0.73 CMA1 (0.35) SMN1; SMN2ALDH1A1AKR1C3AKR1C2KMT2A
SCHEMBL474729 0.73 CMA1 (0.35) SMN1; SMN2ALDH1A1AKR1C3AKR1C2KMT2A
SCHEMBL474976 0.72 PTGDR2 (0.39) SMN1; SMN2ALDH1A1GLAMAPK14PTGS2
SCHEMBL473961 0.72 ALDH1A1 (0.41) SMN1; SMN2ALDH1A1KMT2AMAPTLMNA
SCHEMBL474936 0.71 ADORA2A (0.42) SMN1; SMN2BRPF1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed