SCHEMBL474051

SCHEMBL474051

CC(c1cc(C(=O)O)ccc1-c1ccccc1)C(O)(c1ccc2oc(=O)n(C)c2c1)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
HPGD P15428 1/20 0.39
KMO O15229 1/20 0.36
ASAH1 Q13510 2/20 0.35
CREBBP Q92793 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
S1PR1 P21453 1/20 0.34
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33
HPSE Q9Y251 1/20 0.33
KCNJ1 P48048 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473904 0.94 ALDH1A1 (0.46) ALDH1A1HPGDASAH1MEN1KMT2A
SCHEMBL473917 0.91 ALDH1A1 (0.36) ALDH1A1HPGDKMOASAH1MEN1
SCHEMBL474633 0.85 ALDH1A1 (0.41) ALDH1A1S1PR1PRKAG1PRKAA1PRKAB1
SCHEMBL474061 0.84 KMO (0.38) ALDH1A1HPGDKMOCREBBPMEN1
SCHEMBL473993 0.83 MAPK14 (0.40) ALDH1A1KMOASAH1
SCHEMBL473905 0.82 PSEN1 (0.34) KMOMEN1KMT2ATP53POLB
SCHEMBL12164105 0.82 PSEN1 (0.34) KMOMEN1KMT2ATP53POLB
SCHEMBL474057 0.82 KMO (0.36) ALDH1A1HPGDKMOASAH1MAPT
SCHEMBL473958 0.77 ALDH1A1 (0.37) ALDH1A1POLBTHRB
SCHEMBL473943 0.77 KCNJ1 (0.41) KMOCREBBPTP53POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed