SCHEMBL4747756

SCHEMBL4747756

CCN1CCc2cc(C)nc(-c3ccc(F)cc3)c2C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.39
ADORA2A P29274 4/20 0.37
ADORA1 P30542 3/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
KCNH2 Q12809 1/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CYP19A1 P11511 2/20 0.37
KDM4E B2RXH2 1/20 0.36
NOTUM Q6P988 1/20 0.36
CCNT1 O60563 1/20 0.36
CDK4 P11802 1/20 0.36
CCNA2 P20248 1/20 0.36
CCND1 P24385 1/20 0.36
CDK2 P24941 1/20 0.36
CCND3 P30281 1/20 0.36
CDK7 P50613 1/20 0.36
CDK9 P50750 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4747297 0.87 HRH3 (0.42) HRH3ADORA2AADORA1ALDH1A1HPGD
SCHEMBL4786612 0.86 ALDH1A1 (0.39) HRH3ADORA2AADORA1ALDH1A1HPGD
SCHEMBL4750242 0.85 HRH3 (0.58) HRH3KCNH2
SCHEMBL4750215 0.85 PDGFRB (0.42) HRH3ADORA2AADORA1ALDH1A1HPGD
SCHEMBL4786809 0.85 GAA (0.45) ALDH1A1HPGDGAASMN1; SMN2HSD17B10
SCHEMBL4751106 0.84 GABRG2 (0.41) HRH3ADORA2AADORA1ALDH1A1HPGD
SCHEMBL4747888 0.84 MAPK13 (0.49) HRH3ADORA2AADORA1ALDH1A1HPGD
SCHEMBL4788225 0.82 HRH3 (0.38) HRH3KCNH2
SCHEMBL4788585 0.82 CASP3 (0.43) HRH3ADORA2AADORA1GAA
SCHEMBL4747794 0.82 POLB (0.44) ADORA2AADORA1ALDH1A1KCNH2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed