SCHEMBL4751106

SCHEMBL4751106

Cc1cc2c(c(-c3ccc(F)cc3)n1)C(=O)N(C)CC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
KCNH2 Q12809 1/20 0.41
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
HPGD P15428 2/20 0.40
ADORA2A P29274 6/20 0.39
ADORA1 P30542 5/20 0.39
CSNK1D P48730 2/20 0.38
MAPK9 P45984 2/20 0.38
NUAK1 O60285 1/20 0.38
ROCK2 O75116 1/20 0.38
MAP4K4 O95819 1/20 0.38
LCK P06239 1/20 0.38
MAPK8 P45983 1/20 0.38
CSNK1A1 P48729 1/20 0.38
CSNK1E P49674 1/20 0.38
GSK3B P49841 1/20 0.38
MAP2K1 Q02750 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4747756 0.84 HRH3 (0.39) KCNH2ALDH1A1KDM4EHPGDADORA2A
SCHEMBL4747297 0.83 HRH3 (0.42) GABRG2GABRB3GABRA5KCNH2ALDH1A1
SCHEMBL4785722 0.83 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDADORA2AADORA1
SCHEMBL4750242 0.82 HRH3 (0.58) KCNH2HRH3
SCHEMBL4750215 0.82 PDGFRB (0.42) GABRG2GABRB3GABRA5KCNH2ALDH1A1
SCHEMBL4788529 0.80 HTR2A (0.38) KCNH2ALDH1A1KDM4EADORA2AADORA1
SCHEMBL4786612 0.80 ALDH1A1 (0.39) ALDH1A1HPGDADORA2AADORA1MAPK14
SCHEMBL4747888 0.80 MAPK13 (0.49) ALDH1A1KDM4EHPGDADORA2AADORA1
SCHEMBL4788585 0.79 CASP3 (0.43) ADORA2AADORA1MAPK14NPC1MAPT
SCHEMBL4788225 0.79 HRH3 (0.38) GABRG2GABRB3GABRA5KCNH2MAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO disclosed