SCHEMBL4748040

SCHEMBL4748040

CCOC(=O)C1(Cc2ccncc2)Cc2cc(OC)c(OC)cc2C1=O

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.41
LMNA P02545 1/20 0.41
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 2/20 0.40
PDE4D Q08499 7/20 0.39
PDE4A P27815 3/20 0.39
PDE4B Q07343 3/20 0.39
PDE4C Q08493 3/20 0.39
GAA P10253 1/20 0.38
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5718421 0.90 MAPT (0.42) KDM4ELMNAKMT2AALDH1A1PDE4D
SCHEMBL17320350 0.86 KDM4E (0.39) KDM4ELMNAKMT2AALDH1A1PDE4D
SCHEMBL15906591 0.85 KDM4E (0.38) KDM4ELMNAKMT2AALDH1A1PDE4A
SCHEMBL15899269 0.79 KDM4E (0.36) KDM4ELMNAKMT2AALDH1A1PDE4D
SCHEMBL13988029 0.79 KDM4E (0.45) KDM4ELMNAKMT2AALDH1A1GAA
SCHEMBL13989627 0.77 PDE4D (0.43) KDM4EKMT2AALDH1A1PDE4DPDE4A
SCHEMBL13987170 0.77 KDM4E (0.43) KDM4ELMNAKMT2AALDH1A1GAA
SCHEMBL13987169 0.77 KDM4E (0.43) KDM4ELMNAKMT2AALDH1A1GAA
SCHEMBL9358766 0.76 KDM4E (0.43) KDM4ELMNAKMT2AALDH1A1GAA
SCHEMBL14026620 0.75 PDE4D (0.39) KMT2AALDH1A1PDE4DPDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966136-B1 NOVEL PROCESS FOR PRODUCTION OF HIGHLY PURE POLYMORPH (I) DONEPEZIL HYDROCHLORIDE RICHTER GEDEON NYRT (HU) 2014-02-26 EP disclosed
EP-1954676-B1 PROCESS FOR MAKING DONEPEZIL SYNTHON BV (NL) 2012-11-07 EP disclosed
US-20080306271-A1 Novel Process for Production of Highly Pure Polymorph (I) Donepezil Hydrochloride RICHTER GEDEON NYRT. (HU) 2008-12-11 US disclosed
EP-1966136-A2 NOVEL PROCESS FOR PRODUCTION OF HIGHLY PURE POLYMORPH (I) DONEPEZIL HYDROCHLORIDE Richter Gedeon NYRT (HU) 2008-09-10 EP disclosed
EP-1954676-A2 PROCESS FOR MAKING DONEPEZIL Synthon B.V. (NL) 2008-08-13 EP disclosed
WO-2007072087-A2 NOVEL PROCESS FOR PRODUCTION OF HIGHLY PURE POLYMORPH (I) DONEPEZIL HYDROCHLORIDE RICHTER GEDEON NYRT. (HU) 2007-06-28 WO disclosed
US-20070135644-A1 PROCESS FOR MAKING DONEPEZIL SYNTHON BV (NL) 2007-06-14 US disclosed
WO-2007057226-A2 PROCESS FOR MAKING DONEPEZIL SYNTHON B.V. (NL) 2007-05-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080306271-A1 Novel Process for Production of Highly Pure Polymorph (I) Donepezil Hydrochloride DRD4, IDO1, ADH1A KDM4E 99/4885LMNA 2962/4885KMT2A 412/4885
US-20070135644-A1 PROCESS FOR MAKING DONEPEZIL MAOA, ACHE, CHAT KDM4E 104/4885LMNA 2498/4885KMT2A 24/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.