SCHEMBL4748723

SCHEMBL4748723

O=C(O)c1cc2c(NCc3ccc(OC(F)(F)F)cc3)cccc2n1Cc1cccc(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.51
CCR2 P41597 11/20 0.50
TRPV1 Q8NER1 1/20 0.44
PLA2G2A P14555 2/20 0.44
PTGER4 P35408 1/20 0.44
SERPINE1 P05121 1/20 0.42
EPHX2 P34913 1/20 0.42
PPARA Q07869 1/20 0.42
PPARG P37231 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4650004 0.88 CCR2 (0.54) CCR2PLA2G2A
SCHEMBL4650663 0.87 CCR2 (0.55) CCR2PLA2G2APTGER4
SCHEMBL4650169 0.84 CCR9 (0.55) CCR2
SCHEMBL4648818 0.84 CCR2 (0.53) CCR2PPARG
SCHEMBL4649957 0.83 CCR2 (0.53) CCR2PLA2G2APTGER4
SCHEMBL4807606 0.81 CCR2 (0.51) CCR2PTGER4
SCHEMBL4649909 0.80 CCR2 (0.50) CCR2PTGER4
SCHEMBL4653137 0.78 CCR2 (0.47) CCR2PTGER4PPARG
SCHEMBL4649594 0.77 CCR2 (0.48) PTGESCCR2PPARG
SCHEMBL4652792 0.76 CCR2 (0.49) CCR2PLA2G2APPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904487-A2 INDOLE DERIVATIVES FOR THE TREATMENT OF TUBERCULOSIS AstraZeneca AB (SE) 2008-04-02 EP disclosed
WO-2006067392-A2 INDOLE DERIVATIVES FOR THE TREATMENT OF TUBERCULOSIS ASTRAZENECA AB (SE) 2006-06-29 WO disclosed