SCHEMBL4650004

SCHEMBL4650004

O=C(O)c1cc2c(NCc3ccc(C(F)(F)F)cc3)cccc2n1Cc1cccc(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 13/20 0.54
CCR9 P51686 4/20 0.50
MAPT P10636 1/20 0.43
F10 P00742 1/20 0.43
PLA2G2A P14555 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4648818 0.93 CCR2 (0.53) CCR2CCR9MAPTF10
SCHEMBL4650169 0.91 CCR9 (0.55) CCR2CCR9
SCHEMBL4748723 0.88 PTGES (0.51) CCR2PLA2G2A
SCHEMBL4650663 0.87 CCR2 (0.55) CCR2CCR9MAPTF10PLA2G2A
SCHEMBL4649957 0.86 CCR2 (0.53) CCR2CCR9MAPTF10PLA2G2A
SCHEMBL4649909 0.84 CCR2 (0.50) CCR2MAPTF10
SCHEMBL4807606 0.83 CCR2 (0.51) CCR2MAPTF10
SCHEMBL4653137 0.80 CCR2 (0.47) CCR2MAPTF10
SCHEMBL4649594 0.79 CCR2 (0.48) CCR2MAPTF10
SCHEMBL4649469 0.76 CCR2 (0.55) CCR2MAPTF10PLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904487-A2 INDOLE DERIVATIVES FOR THE TREATMENT OF TUBERCULOSIS AstraZeneca AB (SE) 2008-04-02 EP disclosed
WO-2006067392-A2 INDOLE DERIVATIVES FOR THE TREATMENT OF TUBERCULOSIS ASTRAZENECA AB (SE) 2006-06-29 WO disclosed