SCHEMBL4748892

SCHEMBL4748892

CO[C@H]1CN(C)CCc2cc(C(=O)O)sc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
GLA P06280 1/20 0.37
DAO P14920 1/20 0.37
NOTUM Q6P988 3/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
HPGD P15428 2/20 0.33
LMNA P02545 1/20 0.33
DRD1 P21728 5/20 0.33
MAPK1 P28482 1/20 0.33
THPO P40225 1/20 0.33
HIF1A Q16665 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MTOR P42345 1/20 0.33
TBXAS1 P24557 2/20 0.32
MAPT P10636 1/20 0.32
BLM P54132 1/20 0.32
PMP22 Q01453 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4748891 1.00 KDM4E (0.37) KDM4EALDH1A1GLADAONOTUM
SCHEMBL4751950 0.91 ALDH1A1 (0.40) KDM4EALDH1A1GLACYP3A4HPGD
SCHEMBL3304805 0.83 ALDH1A1 (0.41) KDM4EALDH1A1GLADAONOTUM
SCHEMBL4752664 0.79 ALDH1A1 (0.37) KDM4EALDH1A1GLADAOCYP3A4
SCHEMBL3310259 0.79 ALDH1A1 (0.37) KDM4EALDH1A1GLADAOCYP3A4
SCHEMBL4751943 0.78 DRD1 (0.34) CYP3A4CYP2D6LMNADRD1MAPK1
SCHEMBL3308515 0.77 ALDH1A1 (0.42) KDM4EALDH1A1GLAHPGDLMNA
SCHEMBL3308910 0.73 MAOA (0.43) KDM4EALDH1A1GLADAONOTUM
SCHEMBL3308872 0.73 MAOA (0.43) KDM4EALDH1A1GLADAONOTUM
SCHEMBL3303694 0.73 KDM4E (0.36) KDM4EALDH1A1GLADAONOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135526-A1 CARBOXYLIC ACID AMIDES AS FACTOR XA INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-13 WO claimed
WO-2008135526-A1 CARBOXYLIC ACID AMIDES AS FACTOR XA INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-13 WO disclosed