SCHEMBL4749301

SCHEMBL4749301

CCc1nc(Cl)cc2c1C(=O)OCC2

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
DYRK1A Q13627 1/20 0.32
DYRK2 Q92630 1/20 0.32
DYRK1B Q9Y463 1/20 0.32
PGR P06401 2/20 0.31
MAT2A P31153 1/20 0.31
DHFR P00374 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4064490 0.89 GLP1R (0.34) MAOAMAOB
SCHEMBL4808073 0.82 DYRK1A (0.39) MAOAMAOBDYRK1ADYRK2DYRK1B
SCHEMBL4245511 0.81 MAPT (0.32)
SCHEMBL4067976 0.80 MAOA (0.40) MAOAMAOBDYRK1ADYRK2DYRK1B
SCHEMBL4067369 0.80 MAOA (0.35) MAOAMAOBDYRK1ADYRK2DYRK1B
SCHEMBL4747016 0.77 MAOA (0.34) MAOAMAOBPGR
SCHEMBL4071256 0.72 MAPT (0.36)
SCHEMBL4749586 0.71 DYRK1A (0.35) MAOAMAOBDYRK1AGAA
SCHEMBL4749400 0.71 MAOA (0.35) MAOAMAOBPGRGAA
SCHEMBL4065469 0.71 ALDH1A1 (0.43) MAOAMAOBDYRK1ADYRK2DYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123756-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTON TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO disclosed