SCHEMBL4750077

SCHEMBL4750077

Cc1ccc(NC(=O)c2cccc(CC(C)C#N)c2)cc1C(=O)Nc1cnc(C)c(C)c1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRAF P15056 18/20 0.57
CYP2C9 P11712 5/20 0.51
LCK P06239 2/20 0.47
BTK Q06187 2/20 0.47
KDR P35968 1/20 0.47
MAPK14 Q16539 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4749868 0.87 BRAF (0.67) BRAFCYP2C9LCKBTKKDR
SCHEMBL4750556 0.86 BRAF (0.67) BRAFCYP2C9LCKBTK
SCHEMBL5803018 0.86 BRAF (0.54) BRAFCYP2C9LCKMAPK14
SCHEMBL4970779 0.85 NR1H4 (0.49) BRAFCYP2C9
SCHEMBL5802387 0.84 BRAF (0.45) BRAFCYP2C9LCKBTK
SCHEMBL5799643 0.84 BRAF (0.49) BRAFCYP2C9BTKMAPK14
SCHEMBL5801432 0.83 BRAF (0.52) BRAFCYP2C9LCKBTKKDR
SCHEMBL4966996 0.80 ROCK2 (0.44) BRAFMAPK14
SCHEMBL3934670 0.79 BRAF (0.88) BRAFCYP2C9LCKBTKKDR
SCHEMBL5212609 0.76 MAPT (0.52) CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008120004-A1 COMBINATION OF A MEK- INHIBITOR AND A B-RAF INHIBITOR FOR THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2008-10-09 WO claimed