SCHEMBL4750592

SCHEMBL4750592

C=CC(C)C(C)(N)c1ccc(C(=O)O)c(C)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRB P28702 2/20 0.44
NR1H4 Q96RI1 6/20 0.41
RXRA P19793 1/20 0.40
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
GRIN2C Q14957 1/20 0.34
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2997583 0.75 RXRB (0.46) RXRBNR1H4RXRATDP1ALDH1A1
SCHEMBL2806543 0.72 RXRB (0.59) RXRBNR1H4RXRATDP1ALDH1A1
SCHEMBL30295343 0.72 RXRB (0.59) RXRBNR1H4RXRATDP1ALDH1A1
SCHEMBL162565 0.72 RXRB (0.69) RXRBNR1H4RXRATDP1EPHX2
SCHEMBL17908058 0.71 RXRB (0.57) RXRBNR1H4RXRATDP1ALDH1A1
SCHEMBL838388 0.71 CYP2D6 (0.40) ALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL4896201 0.71 CYP2D6 (0.40) ALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL10048583 0.71 CYP2D6 (0.40) ALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL28191970 0.70 RXRB (0.58) RXRBNR1H4RXRATDP1ALDH1A1
SCHEMBL863182 0.68 ALDH1A1 (0.37) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008119162-A1 METHODS OF PREPARING PRIMARY, SECONDARY AND TERTIARY CARBINAMINE COMPOUNDS IN THE PRESENCE OF AMMONIA KANATA CHEMICAL TECHNOLOGIES INC. (CA) 2008-10-09 WO disclosed