SCHEMBL863182

SCHEMBL863182

C=CC(C)C(C)(N)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
KIF11 P52732 2/20 0.35
ORAI1 Q96D31 1/20 0.35
ORAI2 Q96SN7 1/20 0.35
ORAI3 Q9BRQ5 1/20 0.35
TRPV6 Q9H1D0 1/20 0.35
PDE2A O00408 3/20 0.35
TGM2 P21980 1/20 0.35
NOS1 P29475 1/20 0.35
TAAR1 Q96RJ0 1/20 0.33
TEAD1 P28347 2/20 0.33
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
PLAU P00749 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
IDO1 P14902 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL838387 1.00 ALDH1A1 (0.37) ALDH1A1KIF11ORAI1ORAI2ORAI3
SCHEMBL878960 1.00 ALDH1A1 (0.37) ALDH1A1KIF11ORAI1ORAI2ORAI3
SCHEMBL837837 1.00 ALDH1A1 (0.37) ALDH1A1KIF11ORAI1ORAI2ORAI3
SCHEMBL10048583 0.81 CYP2D6 (0.40) ALDH1A1TAAR1
SCHEMBL4896201 0.81 CYP2D6 (0.40) ALDH1A1TAAR1
SCHEMBL838388 0.81 CYP2D6 (0.40) ALDH1A1TAAR1
SCHEMBL963755 0.70 PDE2A (0.58) ALDH1A1KIF11ORAI1ORAI2ORAI3
SCHEMBL4750592 0.68 RXRB (0.44) ALDH1A1
Hydrochloric Acid SCHEMBL18920592 0.68 PDE2A (0.56) ALDH1A1KIF11ORAI1ORAI2ORAI3
SCHEMBL13246739 0.68 TACR1 (0.41) ALDH1A1KIF11PDE2ATGM2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143451-B2 Reacting a ketone with an allyl boron compound anc ammonia or ammonium salt; synthons KANATA CHEMICAL TECHNOLOGIES INC. (CA) 2012-03-27 US disclosed
US-20080139847-A1 METHODS OF PREPARING TERTIARY CARBINAMINE COMPOUNDS KANATA CHEMICAL TECHNOLOGIES INC. (CA) 2008-06-12 US disclosed
US-20080139847-A1 METHODS OF PREPARING TERTIARY CARBINAMINE COMPOUNDS KANATA CHEMICAL TECHNOLOGIES INC. (CA) 2008-06-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080139847-A1 METHODS OF PREPARING TERTIARY CARBINAMINE COMPOUNDS INMT, CROCC, GNMT ALDH1A1 1599/4885KIF11 1608/4885ORAI1 4783/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.