SCHEMBL4751098

SCHEMBL4751098

CCn1ccc2cc(-c3ccc(F)c(F)c3)nc(C)c2c1=O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 11/20 0.38
KDM1A O60341 1/20 0.35
PKM P14618 1/20 0.34
MAPT P10636 1/20 0.34
GRIN2B Q13224 3/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
GRIN1 Q05586 1/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5816274 0.88 ALDH1A1 (0.43) GRM2MAPTNPC1RAB9AALDH1A1
SCHEMBL5818400 0.84 ZAP70 (0.38) GRM2NPC1RAB9AUSP2ALDH1A1
SCHEMBL4750229 0.82 CYP19A1 (0.45) GRM2MAPTALDH1A1
SCHEMBL4747271 0.79 EGFR (0.37) GRM2NPC1RAB9AUSP2ALDH1A1
SCHEMBL4750210 0.79 EGFR (0.39) NPC1RAB9AUSP2ALDH1A1CYP1A2
SCHEMBL4750004 0.76 GRM2 (0.39) GRM2PKMALDH1A1
SCHEMBL4747315 0.74 EGFR (0.49) MAPTNPC1RAB9AALDH1A1
SCHEMBL4750230 0.73 CYP1A2 (0.38) ALDH1A1CYP1A2CYP3A4
SCHEMBL4747830 0.70 RAD51 (0.42) KDM1AMAPTNPC1RAB9AALDH1A1
SCHEMBL5815996 0.70 ALDH1A1 (0.37) GRM2MAPTNPC1RAB9AUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed
WO-2006112666-A1 PYRIDINE DERIVATIVES, METHODS OF THEIR PREPARATIONS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SK CHEMICALS CO., LTD. (KR) 2006-10-26 WO claimed
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO disclosed
WO-2006112666-A1 PYRIDINE DERIVATIVES, METHODS OF THEIR PREPARATIONS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SK CHEMICALS CO., LTD. (KR) 2006-10-26 WO disclosed