SCHEMBL4750004

SCHEMBL4750004

CCn1ccc2cc(C)nc(C)c2c1=O

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 16/20 0.39
PKM P14618 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4747299 0.84 GRM2 (0.38) GRM2PKMKDM4EALDH1A1MAPK1
SCHEMBL4747263 0.82 GRM2 (0.36) GRM2KDM4EALDH1A1
SCHEMBL4747767 0.80 GRM2 (0.37) GRM2
SCHEMBL4750229 0.80 CYP19A1 (0.45) GRM2KDM4EALDH1A1MAPK1
SCHEMBL5816274 0.78 ALDH1A1 (0.43) GRM2KDM4EALDH1A1MAPK1
SCHEMBL4747715 0.78 PDE2A (0.37) GRM2ALDH1A1
SCHEMBL5815996 0.78 ALDH1A1 (0.37) GRM2KDM4EALDH1A1
SCHEMBL4750217 0.77 PDE2A (0.37) GRM2ALDH1A1
SCHEMBL4751098 0.76 GRM2 (0.38) GRM2PKMALDH1A1
SCHEMBL4750023 0.76 HSF1 (0.41) GRM2PKMKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO disclosed