SCHEMBL4785722

SCHEMBL4785722

Cc1cc2c(c(-c3ccc(F)cc3)n1)C(=O)N(C(=O)O)CC2

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
CYP11B2 P19099 3/20 0.38
CYP11B1 P15538 1/20 0.38
ADORA2A P29274 4/20 0.38
ADORA1 P30542 3/20 0.38
NOTUM Q6P988 1/20 0.38
NAMPT P43490 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
HPGD P15428 1/20 0.35
LMNA P02545 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788529 0.88 HTR2A (0.38) ALDH1A1CYP11B2CYP11B1ADORA2AADORA1
SCHEMBL4786612 0.83 ALDH1A1 (0.39) ALDH1A1ADORA2AADORA1NAMPTHPGD
SCHEMBL4751106 0.83 GABRG2 (0.41) ALDH1A1CYP11B2CYP11B1ADORA2AADORA1
SCHEMBL4747756 0.80 HRH3 (0.39) ALDH1A1ADORA2AADORA1NOTUMKDM4E
SCHEMBL4747297 0.80 HRH3 (0.42) ALDH1A1ADORA2AADORA1NAMPTKDM4E
SCHEMBL4786809 0.78 GAA (0.45) ALDH1A1KDM4EMAPTHPGDNPSR1
SCHEMBL4788585 0.77 CASP3 (0.43) ADORA2AADORA1MAPTRAB9AMEN1
SCHEMBL4750242 0.76 HRH3 (0.58)
SCHEMBL4750215 0.76 PDGFRB (0.42) ALDH1A1ADORA2AADORA1KDM4EMAPT
SCHEMBL4788225 0.75 HRH3 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO disclosed