SCHEMBL4752250

SCHEMBL4752250

COCCn1nc(C2CC2)c(Oc2cc(C)c(C#N)c(C)c2)c1CO

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD2 P25440 3/20 0.33
CREBBP Q92793 2/20 0.33
BRD4 O60885 2/20 0.33
BRD3 Q15059 2/20 0.33
ALDH1A1 P00352 4/20 0.32
KDM4E B2RXH2 3/20 0.32
HPGD P15428 3/20 0.32
HSD17B10 Q99714 3/20 0.32
CASP1 P29466 2/20 0.32
CASP7 P55210 2/20 0.32
GAA P10253 2/20 0.32
MAPT P10636 1/20 0.32
KLK7 P49862 1/20 0.32
HTT P42858 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
LMNA P02545 1/20 0.31
TSHR P16473 1/20 0.31
IDH1 O75874 1/20 0.31
PDE10A Q9Y233 1/20 0.30
PGR P06401 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4748729 0.88 KDM4E (0.32) ALDH1A1KDM4ELMNA
SCHEMBL4752257 0.86 PDE10A (0.34) ALDH1A1KDM4EMAPTSMN1; SMN2LMNA
SCHEMBL4748819 0.83 PGR (0.37) ALDH1A1KDM4ELMNAPGR
SCHEMBL4752262 0.82 ALDH1A1 (0.36) BRD2CREBBPBRD4BRD3ALDH1A1
SCHEMBL4751253 0.82 PGR (0.40) ALDH1A1KDM4ELMNAPGR
SCHEMBL4097765 0.80 KDM4E (0.35) BRD4ALDH1A1KDM4EMAPTLMNA
SCHEMBL4904300 0.80 PGR (0.34) ALDH1A1KDM4ELMNATSHRPGR
SCHEMBL4110176 0.79 KDM4E (0.34) ALDH1A1KDM4EMAPTLMNAPDE10A
SCHEMBL4854390 0.77
SCHEMBL14022484 0.75 KDM4E (0.33) ALDH1A1KDM4EHPGDHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135824-A1 OXYALKYLPYRAZOLE COMPOUNDS USEFUL IN THERAPY PFIZER LIMITED (GB) 2008-11-13 WO disclosed
WO-2008135824-A1 OXYALKYLPYRAZOLE COMPOUNDS USEFUL IN THERAPY PFIZER LIMITED (GB) 2008-11-13 WO disclosed