SCHEMBL4753169

SCHEMBL4753169

COc1cc(C)c(S(=O)(=O)N2CCN(Cc3ccccc3)CC2)c(C)c1C

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.71
MAPT P10636 3/20 0.71
PKM P14618 1/20 0.64
LMNA P02545 2/20 0.57
POLB P06746 2/20 0.56
GAA P10253 2/20 0.56
TSHR P16473 3/20 0.51
KDM4E B2RXH2 2/20 0.50
HTT P42858 2/20 0.49
KMT2A Q03164 2/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
MEN1 O00255 1/20 0.49
GLA P06280 1/20 0.49
TP53 P04637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5093036 0.81 ALDH1A1 (0.50) ALDH1A1MAPTLMNAGAATSHR
SCHEMBL5128261 0.76 EPHX2 (0.47) ALDH1A1MAPTKDM4E
SCHEMBL3926267 0.75 ALDH1A1 (0.47) ALDH1A1MAPTPKMKMT2AMEN1
SCHEMBL5666046 0.75 ALDH1A1 (0.44) ALDH1A1MAPTPKMPOLBGAA
SCHEMBL3917745 0.73 ALDH1A1 (0.43) ALDH1A1MAPTPKMKMT2AMEN1
SCHEMBL5088905 0.72 EPHX2 (0.52) ALDH1A1TSHRKMT2AL3MBTL1MEN1
SCHEMBL13726504 0.72 CRHBP (0.69) ALDH1A1MAPTPKMLMNAPOLB
SCHEMBL7131206 0.71 KDM4E (0.78) ALDH1A1MAPTLMNAPOLBGAA
SCHEMBL19991949 0.71 LMNA (0.73) ALDH1A1LMNAGAATSHRL3MBTL1
SCHEMBL13726176 0.71 LMNA (0.75) ALDH1A1MAPTPKMLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008147864-A2 METHODS OF USING PIPERAZINE COMPOUNDS IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-12-04 WO claimed
WO-2008147864-A2 METHODS OF USING PIPERAZINE COMPOUNDS IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-12-04 WO disclosed