SCHEMBL4753564

SCHEMBL4753564

COC(=O)c1nc(C2CCCC2)[nH]c1-c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 1/20 0.45
FEN1 P39748 1/20 0.45
ERCC4 Q92889 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
KDM4E B2RXH2 4/20 0.42
ALDH1A1 P00352 4/20 0.42
HPGD P15428 3/20 0.42
HSD17B10 Q99714 2/20 0.42
ADORA3 P0DMS8 5/20 0.42
ADORA1 P30542 5/20 0.42
ADORA2A P29274 3/20 0.41
MAPT P10636 3/20 0.41
ADORA2B P29275 2/20 0.41
POLB P06746 1/20 0.41
SLC6A3 Q01959 1/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4749731 0.99 ERCC1 (0.44) ERCC1FEN1ERCC4SMN1; SMN2KDM4E
SCHEMBL4750309 0.99 ERCC1 (0.44) ERCC1FEN1ERCC4SMN1; SMN2KDM4E
SCHEMBL7987871 0.88 RAB9A (0.43) KDM4EALDH1A1HPGDHSD17B10ADORA3
SCHEMBL8963574 0.80 PDE2A (0.42) SMN1; SMN2KDM4EALDH1A1HPGDADORA3
SCHEMBL28582957 0.76 ERCC1 (0.68) ERCC1FEN1ERCC4SMN1; SMN2KDM4E
SCHEMBL7991847 0.75 ADORA1 (0.47) KDM4EALDH1A1HPGDADORA3ADORA1
SCHEMBL4753462 0.74 CYP2D6 (0.40) SMN1; SMN2ALDH1A1HSD17B10ADORA3ADORA2A
SCHEMBL28916010 0.74 ERCC1 (0.64) ERCC1FEN1ERCC4SMN1; SMN2KDM4E
SCHEMBL9517058 0.73 RAF1 (0.62) SMN1; SMN2KDM4EHPGDADORA3ADORA1
SCHEMBL9514583 0.72 RAF1 (0.64) ADORA3ADORA1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008139941-A1 SUBSTITUTED IMIDAZOLE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-20 WO disclosed