SCHEMBL4754375

SCHEMBL4754375

COC(=O)NCCOCCC(NC(C)C)c1cccc(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.43
MAPT P10636 3/20 0.43
TSHR P16473 2/20 0.43
MAPK1 P28482 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
LMNA P02545 3/20 0.43
RAB9A P51151 1/20 0.42
REN P00797 8/20 0.41
CYP3A4 P08684 3/20 0.41
HPGD P15428 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
EPHX2 P34913 1/20 0.38
SLC6A4 P31645 1/20 0.37
CASR P41180 1/20 0.37
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755350 0.90 SLC6A4 (0.40) HTTMAPTTSHRMAPK1MEN1
SCHEMBL4753692 0.89 HTT (0.42) HTTMAPTTSHRMAPK1MEN1
SCHEMBL4756964 0.87 REN (0.41) HTTMAPTTSHRMAPK1MEN1
SCHEMBL4757031 0.86 EPHX2 (0.41) HTTMAPTTSHRMAPK1MEN1
SCHEMBL4754003 0.78 SLC6A4 (0.44) HTTMAPTTSHRMAPK1MEN1
SCHEMBL499635 0.76 REN (0.46) HTTMAPTTSHRMAPK1MEN1
SCHEMBL27752438 0.74 WDR5 (0.50) MAPTMEN1KMT2ARAB9AHPGD
SCHEMBL498922 0.73 SLC6A4 (0.52) HTTMAPTTSHRMAPK1MEN1
SCHEMBL499203 0.73 SLC6A4 (0.52) HTTMAPTTSHRMAPK1MEN1
SCHEMBL14252613 0.72 ADRB2 (0.43) MAPK1HPGDSLC6A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156816-A2 RENIN INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2008-12-24 WO disclosed