SCHEMBL4755013

SCHEMBL4755013

N#Cc1ccc2cc(CCN3CC[CH]C(F)C3)c(=O)[nH]c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.44
IDH1 O75874 4/20 0.41
CHEK1 O14757 3/20 0.40
DRD2 P14416 3/20 0.39
DRD4 P21917 3/20 0.39
DRD3 P35462 3/20 0.39
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
KDM4E B2RXH2 3/20 0.36
HSD17B10 Q99714 3/20 0.36
HRH3 Q9Y5N1 1/20 0.35
HTR1A P08908 1/20 0.35
TP53 P04637 1/20 0.35
HTT P42858 1/20 0.35
CYP1A2 P05177 1/20 0.34
POLB P06746 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4441167 0.85 PARP1 (0.44) PARP1IDH1CHEK1DRD2DRD4
SCHEMBL3846224 0.85 PARP1 (0.46) PARP1IDH1CHEK1DRD2DRD4
SCHEMBL4444391 0.81 TP53 (0.40) PARP1IDH1CHEK1DRD2DRD4
SCHEMBL4438705 0.77 PARP1 (0.41) PARP1IDH1CHEK1DRD2DRD4
SCHEMBL5047724 0.76 DRD2 (0.46) PARP1IDH1CHEK1DRD2DRD4
SCHEMBL3846941 0.69 KCNH2 (0.47) PARP1IDH1ALDH1A1LMNAHPGD
SCHEMBL5047695 0.69 PARP1 (0.38) PARP1DRD2HTR1A
SCHEMBL3716513 0.67 IDH1 (0.50) PARP1IDH1DRD2DRD4DRD3
SCHEMBL23482001 0.66 HRH3 (0.60) CHEK1DRD2DRD4DRD3HRH3
SCHEMBL5047854 0.65 MAPK10 (0.42) PARP1CHEK1HTR1AHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001126-A1 SUBSTITUTED PIPERIDINE DERIVATIVES AND THEIR USE AS ANTIBATERIAL AGENTS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed