SCHEMBL3716513

SCHEMBL3716513

N#Cc1ccc2cc(CC(=O)O)c(=O)[nH]c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 4/20 0.50
KDM4E B2RXH2 5/20 0.45
HSD17B10 Q99714 4/20 0.45
ALDH1A1 P00352 4/20 0.45
PIN1 Q13526 1/20 0.45
EGLN1 Q9GZT9 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.42
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41
TSHR P16473 2/20 0.41
HPGD P15428 1/20 0.41
PARP1 P09874 1/20 0.41
FASN P49327 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
DRD2 P14416 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3719538 0.89 IDH1 (0.50) IDH1KDM4EHSD17B10ALDH1A1PIN1
SCHEMBL3709499 0.84 IDH1 (0.49) IDH1KDM4EHSD17B10ALDH1A1SMN1; SMN2
SCHEMBL6238686 0.81 DRD2 (0.50) IDH1PIN1GRIN1GRIN2BPTGDR2
SCHEMBL5678790 0.76 MAPK1 (0.61) KDM4EHSD17B10ALDH1A1SMN1; SMN2GRIN2D
SCHEMBL30434363 0.76 MAPK1 (0.61) KDM4EHSD17B10ALDH1A1SMN1; SMN2GRIN2D
SCHEMBL3396789 0.76 DAO (0.63) IDH1PIN1FASN
SCHEMBL4659631 0.75 KDM4E (0.61) KDM4EHSD17B10ALDH1A1SMN1; SMN2TSHR
SCHEMBL3718386 0.75 GRIN2D (0.41) IDH1KDM4EHSD17B10ALDH1A1GRIN2D
SCHEMBL327599 0.73 PIN1 (0.55) KDM4EHSD17B10ALDH1A1PIN1TSHR
SCHEMBL30180579 0.73 PIN1 (0.55) KDM4EHSD17B10ALDH1A1PIN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393806-A1 INHIBITORS OF JUN N-TERMINAL KINASE Elan Pharmaceuticals Inc. (US) 2011-12-14 EP disclosed
WO-2010091310-A1 INHIBITORS OF JUN N-TERMINAL KINASE ELAN PHARMACEUTICALS, INC. (US) 2010-08-12 WO disclosed