SCHEMBL4755137

SCHEMBL4755137

CNc1cc(=O)n(-c2ccc(Cl)cc2)c(C2CCC(C(F)(F)F)CC2)n1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 1/20 0.37
MCHR1 Q99705 4/20 0.36
DRD1 P21728 2/20 0.36
DRD5 P21918 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.34
PROKR1 Q8TCW9 3/20 0.33
AOC2 O75106 1/20 0.33
GRM1 Q13255 1/20 0.33
KCNH2 Q12809 1/20 0.33
MAT2A P31153 1/20 0.33
KMT2A Q03164 2/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
MEN1 O00255 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755132 1.00 AVPR1A (0.37) AVPR1AMCHR1DRD1DRD5SMN1; SMN2
Hydrochloric Acid SCHEMBL4822238 0.99 AVPR1A (0.37) AVPR1AMCHR1DRD1DRD5SMN1; SMN2
Hydrochloric Acid SCHEMBL4822247 0.99 AVPR1A (0.37) AVPR1AMCHR1DRD1DRD5SMN1; SMN2
SCHEMBL13985527 0.87 HSD11B1 (0.36) AVPR1AKCNH2
SCHEMBL4755166 0.85 AVPR1A (0.39) AVPR1AMCHR1DRD1DRD5SMN1; SMN2
SCHEMBL4755169 0.85 AVPR1A (0.39) AVPR1AMCHR1DRD1DRD5SMN1; SMN2
SCHEMBL13985298 0.83 BRD4 (0.37) AVPR1ASMN1; SMN2KMT2ACNR1CNR2
SCHEMBL13985222 0.83 AVPR1A (0.39) AVPR1AMCHR1DRD1DRD5SMN1; SMN2
SCHEMBL4789685 0.83 AVPR1A (0.39) AVPR1AMCHR1DRD1DRD5SMN1; SMN2
SCHEMBL4755058 0.83 MCHR1 (0.34) MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO disclosed