SCHEMBL4755218

SCHEMBL4755218

Cc1cc(=O)n(-c2ccc(C#N)nc2)c(C2CCCC(C(F)(F)F)C2)n1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LCAT P04180 1/20 0.35
AR P10275 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4D Q08499 1/20 0.33
USP14 P54578 2/20 0.33
ELANE P08246 1/20 0.33
ADRB1 P08588 1/20 0.33
HTR1A P08908 1/20 0.33
CYP2C9 P11712 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
PIK3CA P42336 1/20 0.31
DPP4 P27487 1/20 0.30
CYP3A4 P08684 1/20 0.30
ERG P11308 1/20 0.30
GPBAR1 Q8TDU6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13985513 1.00 LCAT (0.35) LCATARPDE4BPDE4DUSP14
SCHEMBL13985505 0.82 MCHR1 (0.35) HRH3
SCHEMBL4790013 0.82 MCHR1 (0.35) HRH3
SCHEMBL13985419 0.81 PDE4B (0.34) LCATARPDE4BPDE4DUSP14
SCHEMBL4755607 0.77 PDE4B (0.34) LCATARPDE4BPDE4DUSP14
SCHEMBL13985423 0.77 PDE4B (0.34) LCATARPDE4BPDE4DUSP14
SCHEMBL4755767 0.75 CHRNB2 (0.34) USP14PIK3CA
SCHEMBL4755765 0.75 CHRNB2 (0.34) USP14PIK3CA
SCHEMBL4789984 0.75 KCNH2 (0.32) LCATCYP3A4ERGGPBAR1
SCHEMBL4755652 0.75 PDE4B (0.35) LCATPDE4BPDE4DUSP14PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO disclosed