SCHEMBL4789984

SCHEMBL4789984

Cc1cc(=O)n(-c2cnc(C#N)nc2)c(C2CCC(C(F)(F)F)CC2)n1

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.32
GPR119 Q8TDV5 2/20 0.32
CTSL P07711 1/20 0.32
LCAT P04180 1/20 0.32
PDE1A P54750 1/20 0.32
PDE1B Q01064 1/20 0.32
PDE1C Q14123 1/20 0.32
SPR P35270 2/20 0.31
CYP3A4 P08684 1/20 0.31
ERG P11308 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755651 0.86 SPR (0.32) PDE1APDE1BPDE1CSPR
SCHEMBL13985520 0.84 USP14 (0.38) KCNH2
SCHEMBL4755767 0.81 CHRNB2 (0.34) SPR
SCHEMBL4755765 0.81 CHRNB2 (0.34) SPR
SCHEMBL4755215 0.80 DRD1 (0.40) CYP3A4
SCHEMBL4755592 0.80 DRD1 (0.37)
SCHEMBL4755213 0.80 DRD1 (0.40) CYP3A4
SCHEMBL4755594 0.80 DRD1 (0.37)
SCHEMBL4755659 0.79 MEN1 (0.39)
SCHEMBL4755656 0.79 MEN1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO disclosed