SCHEMBL4755583

SCHEMBL4755583

NC(=O)c1c(C(Cl)(Cl)Cl)nsc1N

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.38
PDGFRB P09619 2/20 0.36
HSD17B10 Q99714 2/20 0.31
KDM4E B2RXH2 2/20 0.30
ALDH1A1 P00352 2/20 0.30
MAPT P10636 2/20 0.30
USP2 O75604 1/20 0.30
HPGD P15428 1/20 0.30
MEN1 O00255 1/20 0.30
RECQL P46063 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4754963 0.81 KDR (0.39) KDRPDGFRBHSD17B10KDM4EALDH1A1
SCHEMBL10500542 0.71 KDR (0.43) KDRPDGFRBHSD17B10KDM4EALDH1A1
SCHEMBL3863859 0.69 KDR (0.45) KDRPDGFRBHSD17B10KDM4EALDH1A1
SCHEMBL18955834 0.65 KDR (0.58) KDRPDGFRBMEN1KMT2A
SCHEMBL15069721 0.63 KDR (0.64) KDRPDGFRBKDM4EALDH1A1MEN1
SCHEMBL4755614 0.63 MEN1 (0.35) ALDH1A1MAPTMEN1KMT2A
SCHEMBL4758106 0.61 CISD2 (0.39) HSD17B10KDM4EALDH1A1MAPTHPGD
SCHEMBL12894820 0.60 KDR (0.35) KDRPDGFRBALDH1A1MAPTHPGD
SCHEMBL3084536 0.60 ALDH1A1 (0.39) KDRPDGFRBHSD17B10ALDH1A1MAPT
SCHEMBL8188239 0.57 KDM4E (0.40) KDRPDGFRBHSD17B10KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001214-A2 THIENO[2,3-D]PYRIMIDIN-4(3H)-ONE, ISOXAZOLO[5,4-D]PYRIMIDIN-4(5H)-ONE AND ISOTHIAZOLO[5,4-D]PYRIMIDIN-4(5H)-ONE DERIVATIVES AS CALCIUM RECEPTOR ANTAGONISTS PFIZER PRODUCTS INC. (US) 2008-12-31 WO disclosed
WO-2009001214-A2 THIENO[2,3-D]PYRIMIDIN-4(3H)-ONE, ISOXAZOLO[5,4-D]PYRIMIDIN-4(5H)-ONE AND ISOTHIAZOLO[5,4-D]PYRIMIDIN-4(5H)-ONE DERIVATIVES AS CALCIUM RECEPTOR ANTAGONISTS PFIZER PRODUCTS INC. (US) 2008-12-31 WO disclosed
WO-2009002106-A2 ANTI-CANCER COMPOSITION COMPRISING AQUATIC MICROBIAL EXTRACT AJOU UNIVERSITY INDUSTRY-ACADEMIC COOPERATION FOUNDATION (KR) 2008-12-31 WO disclosed