SCHEMBL4757644

SCHEMBL4757644

CC1CN(S(=O)(=O)c2c(C(=O)O)n(S(=O)(=O)c3ccccc3)c3ccc(Cl)cc23)C[C@H](C)O1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACLY P53396 2/20 0.51
HTR6 P50406 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PPARG P37231 3/20 0.39
PPARA Q07869 3/20 0.39
PPARD Q03181 2/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
TSHR P16473 1/20 0.39
CXCR2 P25025 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2930564 1.00 ACLY (0.51) ACLYHTR6SMN1; SMN2ALDH1A1TP53
SCHEMBL2930565 1.00 ACLY (0.51) ACLYHTR6SMN1; SMN2ALDH1A1TP53
SCHEMBL2929510 0.88 GAA (0.45) ACLYHTR6SMN1; SMN2ALDH1A1PTGDR2
SCHEMBL2927961 0.88 GAA (0.45) ACLYHTR6SMN1; SMN2ALDH1A1PTGDR2
SCHEMBL2927960 0.88 GAA (0.45) ACLYHTR6SMN1; SMN2ALDH1A1PTGDR2
SCHEMBL4759367 0.83 ACLY (0.53) ACLYHTR6SMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL4757349 0.81 CXCR2 (0.45) ACLYSMN1; SMN2ALDH1A1TP53L3MBTL1
SCHEMBL5823347 0.80 ACLY (0.62) ACLYHTR6PPARGPPARAPPARD
SCHEMBL4757347 0.79 TDP1 (0.42) SMN1; SMN2ALDH1A1TP53L3MBTL1PTGDR2
SCHEMBL2928718 0.77 ACLY (0.55) ACLYPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534695-A4 TYROSINE KINASE INHIBITORS MERCK & CO INC (US) 2008-06-11 EP disclosed
EP-1534695-A2 TYROSINE KINASE INHIBITORS Merck & Co., Inc. (US) 2005-06-01 EP disclosed
WO-2004014851-A2 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2004-02-19 WO disclosed