SCHEMBL4757347

SCHEMBL4757347

CC1CN(S(=O)(=O)c2c(C(=O)OCl)n(S(=O)(=O)c3ccccc3)c3ccccc23)CC(C)O1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.42
ALDH1A1 P00352 3/20 0.41
TP53 P04637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KMT2A Q03164 2/20 0.39
MAPT P10636 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.37
RXFP1 Q9HBX9 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
CXCR2 P25025 1/20 0.37
NPC1 O15118 1/20 0.37
USP2 O75604 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
PKM P14618 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2927960 0.80 GAA (0.45) TDP1ALDH1A1KMT2AMAPTSMN1; SMN2
SCHEMBL2927961 0.80 GAA (0.45) TDP1ALDH1A1KMT2AMAPTSMN1; SMN2
SCHEMBL2929510 0.80 GAA (0.45) TDP1ALDH1A1KMT2AMAPTSMN1; SMN2
SCHEMBL2930564 0.79 ACLY (0.51) TDP1ALDH1A1TP53L3MBTL1SMN1; SMN2
SCHEMBL4757644 0.79 ACLY (0.51) TDP1ALDH1A1TP53L3MBTL1SMN1; SMN2
SCHEMBL2930565 0.79 ACLY (0.51) TDP1ALDH1A1TP53L3MBTL1SMN1; SMN2
SCHEMBL13765391 0.78 ALDH1A1 (0.43) ALDH1A1KMT2AMAPTSMN1; SMN2GAA
SCHEMBL4757349 0.76 CXCR2 (0.45) TDP1ALDH1A1TP53L3MBTL1MAPT
SCHEMBL13765375 0.70 MEN1 (0.45) ALDH1A1KMT2AMAPTSMN1; SMN2
SCHEMBL12392496 0.69 NOD2 (0.48) ALDH1A1L3MBTL1KMT2AMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534695-A4 TYROSINE KINASE INHIBITORS MERCK & CO INC (US) 2008-06-11 EP disclosed
EP-1534695-A2 TYROSINE KINASE INHIBITORS Merck & Co., Inc. (US) 2005-06-01 EP disclosed
WO-2004014851-A2 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2004-02-19 WO disclosed