SCHEMBL4758236

SCHEMBL4758236

CCOC(=O)CC(=O)NNC(=O)c1cc(Cl)cc(N2CCC(O[Si](C)(C)C(C)(C)C)C2)c1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DDR1 Q08345 7/20 0.34
CACNA1I Q9P0X4 6/20 0.34
KCNH2 Q12809 4/20 0.34
ACACB O00763 2/20 0.33
CACNA1G O43497 1/20 0.33
CHRM2 P08172 1/20 0.33
HRH1 P35367 1/20 0.33
HTR4 Q13639 1/20 0.33
CACNA1C Q13936 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
NOTUM Q6P988 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4758264 0.82 WDR91 (0.40) DDR1KDM4EHRH3NOTUM
SCHEMBL4755128 0.77 MAPK14 (0.44) DDR1KCNH2KDM4E
SCHEMBL4757779 0.76 HDAC3 (0.44) DDR1
SCHEMBL4758284 0.68 SMN1; SMN2 (0.47)
SCHEMBL21430984 0.68 JAK3 (0.37) KDM4E
SCHEMBL4755723 0.66 CSF1R (0.48) DDR1KDM4E
SCHEMBL30461098 0.65 HCRTR1 (0.42) KDM4EHRH3
SCHEMBL7082922 0.65 ACACB (0.43) ACACB
SCHEMBL30807534 0.64 GPR119 (0.39) ACACB
SCHEMBL26760872 0.64 LIPG (0.36) ACACBNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed