SCHEMBL4758705

SCHEMBL4758705

C=CC(=O)N1C[C@H](C[C@@](C)(OC(N)=O)c2cccc3ccccc23)[C@@H](c2ccccc2)C1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 7/20 0.39
RORC P51449 6/20 0.36
ACHE P22303 1/20 0.34
KRAS P01116 3/20 0.33
TEAD1 P28347 1/20 0.32
TEAD3 Q99594 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
RIPK1 Q13546 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4758707 0.76 CCR5 (0.39) CCR5RORCACHEKRASTEAD1
SCHEMBL3573543 0.72 AOC3 (0.33) CCR5RORC
SCHEMBL4105648 0.70 CCR5 (0.40) CCR5RORCACHEKRAS
SCHEMBL4108105 0.69 CCR5 (0.41) CCR5RORC
SCHEMBL4108104 0.69 CCR5 (0.41) CCR5RORC
SCHEMBL4758708 0.69 SSTR4 (0.41) CCR5
SCHEMBL9137874 0.69 PPARG (0.40)
SCHEMBL17351745 0.64 CA2 (0.42)
SCHEMBL11570039 0.63 KDM4E (0.44)
SCHEMBL27944402 0.63 CCR5 (0.49) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1882684-A1 PYRROLIDINE DERIVATIVE OR SALT THEREOF Astellas Pharma Inc. (JP) 2008-01-30 EP disclosed