SCHEMBL476130

SCHEMBL476130

CC(C)(C)C(Cc1ccc(C(F)(F)F)nc1)OC(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 2/20 0.42
KCNQ3 O43525 1/20 0.39
KCNQ2 O43526 1/20 0.39
KCNQ4 P56696 1/20 0.39
KCNQ5 Q9NR82 1/20 0.39
DAO P14920 3/20 0.37
TKT P29401 1/20 0.37
CYP2C8 P10632 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36
MGLL Q99685 1/20 0.36
CSF1R P07333 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP3A5 P20815 1/20 0.35
PPARA Q07869 1/20 0.35
TRPV3 Q8NET8 2/20 0.35
LGMN Q99538 1/20 0.35
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4853164 0.77 DAO (0.41) PPARDKCNQ3KCNQ2KCNQ4KCNQ5
SCHEMBL28474974 0.76 CA2 (0.47)
SCHEMBL1936444 0.75 PPARG (0.41) PPARA
SCHEMBL1937035 0.75 EPHX2 (0.37) CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL4445933 0.74 ALDH1A1 (0.45) PPARDKCNQ3KCNQ2KCNQ4KCNQ5
SCHEMBL4072985 0.74 MME (0.43) PPARA
SCHEMBL28652308 0.73 SRR (0.45) PPARA
SCHEMBL25255517 0.72 GRB2 (0.54) MRGPRX4
SCHEMBL18256345 0.72 GRB2 (0.54) MRGPRX4
SCHEMBL31754268 0.72 GRB2 (0.54) MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2410858-A1 P2X3 RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN Merck Sharp & Dohme Corp. (US) 2012-02-01 EP disclosed