SCHEMBL4761946

SCHEMBL4761946

COc1ccc2oc(C(=O)NC(CC(C)C)C(=O)N(C(=O)Nc3ccccc3F)[C@H]3CCCNCC3=O)cc2c1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 14/20 0.50
TAS1R1 Q7RTX1 14/20 0.50
CTSK P43235 4/20 0.39
CTSL P07711 2/20 0.37
CTSS P25774 2/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CTSB P07858 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4770801 0.86 TAS1R3 (0.49) TAS1R3TAS1R1CTSKCTSLCTSS
SCHEMBL4770805 0.86 TAS1R3 (0.49) TAS1R3TAS1R1CTSKCTSLCTSS
SCHEMBL4765540 0.83 NPC1 (0.37) TAS1R3TAS1R1CTSKCTSLCTSS
SCHEMBL4763005 0.81 TAS1R3 (0.48) TAS1R3TAS1R1CTSKCTSSCTSB
SCHEMBL4770834 0.81 TAS1R3 (0.51) TAS1R3TAS1R1CTSKCTSLCTSS
SCHEMBL4770836 0.81 TAS1R3 (0.51) TAS1R3TAS1R1CTSKCTSLCTSS
SCHEMBL6605727 0.80 NPC1 (0.37) ALDH1A1NPC1
SCHEMBL7425840 0.80 TAS1R3 (0.48) TAS1R3TAS1R1CTSKCTSLCTSS
SCHEMBL4762072 0.80 TAS1R3 (0.49) TAS1R3TAS1R1CTSKCTSLCTSS
SCHEMBL7426728 0.79 TAS1R3 (0.47) TAS1R3TAS1R1CTSKCTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1320370-A4 METHOD OF TREATMENT SMITHKLINE BEECHAM CORP (US) 2008-10-22 EP disclosed
EP-1320370-A1 METHOD OF TREATMENT SmithKline Beecham Corporation (US) 2003-06-25 EP disclosed
WO-2002017924-A1 METHOD OF TREATMENT SMITHKLINE BEECHAM CORPORATION (GB) 2002-03-07 WO disclosed