SCHEMBL4763005

SCHEMBL4763005

CC(C)CC(NC(=O)c1cc2ccccc2s1)C(=O)N(C(=O)Nc1ccccc1F)[C@H]1CCCNCC1=O

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.48
TAS1R1 Q7RTX1 2/20 0.48
CTSK P43235 6/20 0.47
UTS2R Q9UKP6 4/20 0.40
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
OPRM1 P35372 2/20 0.37
NPC1 O15118 1/20 0.37
TRPV4 Q9HBA0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4768735 0.90 CTSK (0.36) TAS1R3TAS1R1CTSKUTS2RNPC1
SCHEMBL4765349 0.84 CTSK (0.46) TAS1R3TAS1R1CTSKUTS2RCTSB
SCHEMBL4765345 0.84 CTSK (0.46) TAS1R3TAS1R1CTSKUTS2RCTSB
SCHEMBL4766646 0.83 CTSK (0.45) CTSKUTS2RCTSBCTSSNPC1
SCHEMBL6771256 0.82 CTSK (0.50) TAS1R3TAS1R1CTSKUTS2RCTSB
SCHEMBL4765540 0.82 NPC1 (0.37) TAS1R3TAS1R1CTSKCTSBCTSS
SCHEMBL4761946 0.81 TAS1R3 (0.50) TAS1R3TAS1R1CTSKCTSBCTSS
SCHEMBL6765735 0.81 CTSK (0.46) TAS1R3TAS1R1CTSKUTS2RCTSB
SCHEMBL4838791 0.81 CTSK (0.46) TAS1R3TAS1R1CTSKUTS2RCTSB
SCHEMBL7037396 0.81 NPC1 (0.39) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1320370-A4 METHOD OF TREATMENT SMITHKLINE BEECHAM CORP (US) 2008-10-22 EP disclosed
EP-1320370-A1 METHOD OF TREATMENT SmithKline Beecham Corporation (US) 2003-06-25 EP disclosed
WO-2002017924-A1 METHOD OF TREATMENT SMITHKLINE BEECHAM CORPORATION (GB) 2002-03-07 WO disclosed