SCHEMBL4762153

SCHEMBL4762153

FC(F)(F)C1NCCc2[nH]cnc21

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.51
LMNA P02545 1/20 0.49
ALDH1A1 P00352 1/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4004258 0.73 RAB9A (0.56) RAB9ALMNAALDH1A1POLB
Hydrochloric Acid SCHEMBL7529821 0.71 RAB9A (0.54) RAB9ALMNAALDH1A1POLB
Hydrochloric Acid SCHEMBL1978418 0.68 RAB9A (0.50) RAB9ALMNAALDH1A1POLB
SCHEMBL3441643 0.68 RAB9A (1.00) RAB9ALMNAALDH1A1POLB
Hydrochloric Acid SCHEMBL11516807 0.68 RAB9A (0.50) RAB9ALMNAALDH1A1POLB
Hydrochloric Acid SCHEMBL9866849 0.67 RAB9A (0.53) RAB9ALMNAALDH1A1POLB
SCHEMBL4357488 0.67 RAB9A (0.74) RAB9ALMNAALDH1A1POLB
SCHEMBL11516141 0.67 RAB9A (0.49) RAB9ALMNAALDH1A1POLB
SCHEMBL6420028 0.66 RAB9A (0.44) RAB9ALMNAALDH1A1POLB
SCHEMBL1991375 0.65 RAB9A (0.66) RAB9ALMNAALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12247027-B2 P2X7 modulators JANSSEN PHARMACEUTICA NV (BE) 2025-03-11 US disclosed
US-20240116930-A1 P2X7 MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2024-04-11 US disclosed
US-11820770-B2 P2X7 modulators JANSSEN PHARMACEUTICA NV (BE) 2023-11-21 US disclosed
US-11820770-B2 P2X7 modulators JANSSEN PHARMACEUTICA NV (BE) 2023-11-21 US disclosed
US-11820770-B2 P2X7 modulators JANSSEN PHARMACEUTICA NV (BE) 2023-11-21 US disclosed
US-20220213095-A1 P2X7 MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2022-07-07 US disclosed
US-20220213095-A1 P2X7 MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2022-07-07 US disclosed
US-11225478-B2 P2X7 modulators JANSSEN PHARMACEUTICA NV (BE) 2022-01-18 US disclosed
US-20200325138-A1 P2X7 Modulators JANSSEN PHARMACEUTICA NV (BE) 2020-10-15 US disclosed
US-10703749-B2 P2X7 modulators JANSSEN PHARMACEUTICA NV (BE) 2020-07-07 US disclosed
US-20140275015-A1 P2X7 MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2014-09-18 US disclosed
US-20140275015-A1 P2X7 MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2014-09-18 US disclosed
EP-1589969-A4 3-AMINO-4-PHENYLBUTANOIC ACID DERIVATIVES AS DIPEPTIDYL PEPTIDASE INHIBITORS FOR THE TREATMENT OR PREVENTION OF DIABETES MERCK & CO INC (US) 2008-08-13 EP disclosed
US-7265128-B2 3-amino-4-phenylbutanoic acid derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes MERCK & CO., INC. (US) 2007-09-04 US disclosed
US-20060069116-A1 3-Amino-4-phenylbutanoic acid derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes MERCK SHARP & DOHME LLC 2006-03-30 US disclosed
EP-1589969-A2 3-AMINO-4-PHENYLBUTANOIC ACID DERIVATIVES AS DIPEPTIDYL PEPTIDASE INHIBITORS FOR THE TREATMENT OR PREVENTION OF DIABETES Merck & Co. Inc. (US) 2005-11-02 EP disclosed
US-6908926-B1 Substituted imidazoles, their preparation and use NOVO NORDISK A/S (DK) 2005-06-21 US disclosed
WO-2004064778-A2 3-AMINO-4-PHENYLBUTANOIC ACID DERIVATIVES AS DIPEPTIDYL PEPTIDASE INHIBITORS FOR THE TREATMENT OR PREVENTION OF DIABETES MERCK & CO. INC. (US) 2004-08-05 WO disclosed
EP-1173438-A1 SUBSTITUTED IMIDAZOLES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 2002-01-23 EP disclosed
WO-2000063208-A1 SUBSTITUTED IMIDAZOLES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 2000-10-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200325138-A1 P2X7 Modulators P2RX2, P2RX7, P2RY2 RAB9A 3242/4885LMNA 2272/4885ALDH1A1 1628/4885
US-12247027-B2 P2X7 modulators P2RX2, P2RX7, P2RY2 RAB9A 3242/4885LMNA 2272/4885ALDH1A1 1628/4885
US-11225478-B2 P2X7 modulators P2RX2, P2RX7, P2RY2 RAB9A 3242/4885LMNA 2272/4885ALDH1A1 1628/4885
US-20060069116-A1 3-Amino-4-phenylbutanoic acid derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes DPP4, DPP3, DPP7 RAB9A 4575/4885LMNA 3093/4885ALDH1A1 686/4885
US-11820770-B2 P2X7 modulators P2RX2, P2RX7, P2RY2 RAB9A 3242/4885LMNA 2272/4885ALDH1A1 1628/4885
US-20220213095-A1 P2X7 MODULATORS P2RX2, P2RX7, P2RY2 RAB9A 3242/4885LMNA 2272/4885ALDH1A1 1628/4885
US-20240116930-A1 P2X7 MODULATORS P2RX2, P2RX7, P2RY2 RAB9A 3242/4885LMNA 2272/4885ALDH1A1 1628/4885
US-10703749-B2 P2X7 modulators P2RX2, P2RX7, P2RY2 RAB9A 3242/4885LMNA 2272/4885ALDH1A1 1628/4885
US-20140275015-A1 P2X7 MODULATORS P2RX2, P2RX7, P2RY2 RAB9A 3242/4885LMNA 2272/4885ALDH1A1 1628/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.