SCHEMBL4763259

SCHEMBL4763259

C[C@@H](CCNC(=O)O)CC(=O)N(Cc1ccccc1)C1CCCNCC1O

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.44
SLC6A2 P23975 13/20 0.38
SLC6A4 P31645 13/20 0.38
SLC18A3 Q16572 1/20 0.36
SLC6A3 Q01959 8/20 0.35
KCNH2 Q12809 2/20 0.35
CYP2D6 P10635 1/20 0.35
GHSR Q92847 1/20 0.34
UBE2M P61081 2/20 0.33
DCUN1D1 Q96GG9 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4765027 0.84 CTSD (0.45) CTSDSLC6A2SLC6A4SLC18A3SLC6A3
SCHEMBL6214947 0.76 CTSD (0.37) CTSDSLC6A2SLC6A4SLC6A3MEN1
SCHEMBL4763254 0.75 CTSD (0.38) CTSDSLC6A2SLC6A4SLC18A3SLC6A3
SCHEMBL4763258 0.75 CTSD (0.38) CTSDSLC6A2SLC6A4SLC18A3SLC6A3
SCHEMBL3956518 0.72 CYP2C9 (0.33) CYP2D6ALDH1A1
SCHEMBL2776534 0.72 CTSD (0.55) CTSDSLC6A2SLC6A4SLC18A3SLC6A3
SCHEMBL2776529 0.72 CTSD (0.55) CTSDSLC6A2SLC6A4SLC18A3SLC6A3
SCHEMBL4765023 0.71 CTSD (0.38) CTSDSLC6A2SLC6A4SLC18A3SLC6A3
SCHEMBL7427599 0.70 MEN1 (0.46) MEN1KMT2AALDH1A1HTT
SCHEMBL5143426 0.69 CTSD (0.55) CTSDSLC6A2SLC6A4SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1320370-A4 METHOD OF TREATMENT SMITHKLINE BEECHAM CORP (US) 2008-10-22 EP disclosed
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1320370-A1 METHOD OF TREATMENT SmithKline Beecham Corporation (US) 2003-06-25 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
WO-2002017924-A1 METHOD OF TREATMENT SMITHKLINE BEECHAM CORPORATION (GB) 2002-03-07 WO disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed