SCHEMBL4763258

SCHEMBL4763258

CC(C)CC(NC(=O)O)C(=O)N(Cc1ccccc1)C1CCCNC[C@@H]1O

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.38
SLC6A2 P23975 7/20 0.38
SLC6A4 P31645 7/20 0.38
SLC6A3 Q01959 3/20 0.38
KCNH2 Q12809 2/20 0.38
CYP2D6 P10635 1/20 0.38
SLC18A3 Q16572 1/20 0.37
GHSR Q92847 1/20 0.37
CTSK P43235 5/20 0.36
CTSL P07711 2/20 0.36
CTSB P07858 2/20 0.36
CTSS P25774 2/20 0.36
CACNA1B Q00975 1/20 0.35
PSMB5 P28074 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4763254 1.00 CTSD (0.38) CTSDSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6590880 0.80 CTSK (0.37) SLC6A2SLC6A4KCNH2CTSKCTSL
SCHEMBL7426317 0.77 CTSK (0.37) KCNH2CTSKCTSLCTSBCTSS
SCHEMBL4763259 0.75 CTSD (0.44) CTSDSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6214945 0.75 MAPK1 (0.44) CTSS
SCHEMBL6611358 0.74 MAPK1 (0.36) PSMB5
SCHEMBL4765027 0.74 CTSD (0.45) CTSDSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL2776529 0.73 CTSD (0.55) CTSDSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL2776534 0.73 CTSD (0.55) CTSDSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4765023 0.72 CTSD (0.38) CTSDSLC6A2SLC6A4SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1320370-A4 METHOD OF TREATMENT SMITHKLINE BEECHAM CORP (US) 2008-10-22 EP disclosed
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1320370-A1 METHOD OF TREATMENT SmithKline Beecham Corporation (US) 2003-06-25 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
WO-2002017924-A1 METHOD OF TREATMENT SMITHKLINE BEECHAM CORPORATION (GB) 2002-03-07 WO disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed